CCG-224406 | GRK2 inhibitor |Probechem Biochemicals

Chemical Structure : CCG-224406

CCG-224406 (CCG 224406;CCG224406)

Catalog No.: PC-70119Not For Human Use, Lab Use Only.

CCG-224406 (CCG224406) is a highly selective and potent GRK2 (G protein-coupled receptor kinase 2) inhibitor with IC50 of 130 nM.M.

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Biological Activity

CCG-224406 (CCG224406) is a highly selective and potent GRK2 (G protein-coupled receptor kinase 2) inhibitor with IC50 of 130 nM.
CCG-224406 displays >700-fold selectivity over other GRK subfamilies, and no detectable inhibition of ROCK1.

Physicochemical Properties

M.Wt	558.57
Formula	C29H27FN6O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(3-((2,6-dimethoxybenzyl)carbamoyl)-4-fluorophenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide

References

1. Waldschmidt HV, et al. J Med Chem. 2016 Apr 28;59(8):3793-807.

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CCG-224406 (CCG 224406;CCG224406)

Biological Activity

Physicochemical Properties

References

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