CCG258208

Chemical Structure : CCG258208

Catalog No.: PC-23974Not For Human Use, Lab Use Only.

CCG258208 is a potent selective GRK2 inhibitor with IC50 of 30 nM, >200-fold selectivity over GRK1 and GRK5.

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Biological Activity

CCG258208 is a potent selective GRK2 inhibitor with IC50 of 30 nM, >200-fold selectivity over GRK1 and GRK5.

M.Wt	452.49
Formula	C24H25FN4O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Benzamide, 5-[(3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-piperidinyl]-2-fluoro-N-(1H-pyrazol-3-ylmethyl)-

1. Bouley RA, et al. Mol Pharmacol. 2020 Jun;97(6):392-401.