Chemical Structure : EF-1502
Catalog No.: PC-26893Not For Human Use, Lab Use Only.
EF-1502 (EF1502) is a selective inhibitor of GABA transporter GAT-1/BGT-1, noncompetitively inhibits both mGAT1 and the betaine/GABA transporter mGAT2 (BGT-1)) with Ki of 4 uM and 5 uM respectively, is inactive at GAT3 and GAT4.
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EF-1502 (EF1502) is a selective inhibitor of GABA transporter GAT-1/BGT-1, noncompetitively inhibits both mGAT1 and the betaine/GABA transporter mGAT2 (BGT-1)) with Ki of 4 uM and 5 uM respectively, is inactive at GAT3 and GAT4.
| M.Wt | 414.58 | |
| Formula | C22H26N2O2S2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. White HS, et al. J Pharmacol Exp Ther. 2005 Feb;312(2):866-74.

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