You are here:Home-Chemical Inhibitors & Agonists-GPCR-Angiotensin Receptor-Azilsartan medoxomil
Azilsartan medoxomil

Chemical Structure : Azilsartan medoxomil

CAS No.: 863031-21-4

Azilsartan medoxomil (TAK 491;TAK-491;TAK491)

Catalog No.: PC-44046Not For Human Use, Lab Use Only.

A specific and potent angiotensin II type 1 receptor (AT1) antagonist with IC50 of 2.6 nM, used in the treatment of adults with essential hypertension. .

Packing Price Stock Quantity
10 mg $120 In stock
50 mg $360 In stock
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

A specific and potent angiotensin II type 1 receptor (AT1) antagonist with IC50 of 2.6 nM, used in the treatment of adults with essential hypertension.

Hypertension

Approved

Physicochemical Properties

M.Wt 568.5336
Formula C30H24N4O8
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

1H-Benzimidazole-7-carboxylic acid, 1-[[2'-(2,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-, (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl ester

References

1. French C, et al. J Cardiovasc Pharmacol. 2011 Aug;58(2):143-8.

2. Kusumoto K, et al. Eur J Pharmacol. 2011 Nov 1;669(1-3):84-93.

3. Bönner G, et al. J Hum Hypertens. 2013 Aug;27(8):479-86.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: