DCP1-3

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Chemical Structure : DCP1-3

Catalog No.: PC-72732Not For Human Use, Lab Use Only.

DCP1-3 is a novel allosteric ligand of the angiotensin receptor AT1R, displays NAM potency on AngIV with IC50 of 0.29 uM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

DCP1-3 is a novel allosteric ligand of the angiotensin receptor AT1R, displays NAM potency on AngIV with IC50 of 0.29 uM.
DCP1-3 reduces AngII-induced contraction in renal and iliac arteries in mice.
DCP1-3 inhibits IgG binding to HEK-AT1R cells with IC50 of 2.9 nM.
DCP1-3 reverses PAM effect of the IgG on the agonist-induced calcium response.

Physicochemical Properties

M.Wt	396.459
Formula	C20H29FN2O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-((1R,2R,3R,4R)-4-(3-fluorophenoxy)-3-hydroxy-2-((2-hydroxyethyl)(methyl)amino)cyclopentyl)tetrahydro-2H-pyran-4-carboxamide

References

1. Singh KD, et al. Proc Natl Acad Sci U S A. 2021 Aug 17;118(33):e2019126118.

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DCP1-3

Biological Activity

Physicochemical Properties

References

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