Chemical Structure : 4E2RCat
CAS No.:
432499-63-3
4E2RCat
(eIF4E-eIF4G inhibitor)
Catalog No. : PC-42237Not For Human Use, Lab Use Only.
4E2RCat is a small molecule inhibitor of eIF4E-eIF4G interaction with IC50 of 13.5 uM in TR-FRET-based assay.
Packing Price Stock Quantity 5 mg $168 In stock 0 1 2 3 4 5 10 mg $238 In stock 0 1 2 3 4 5 25 mg $398 In stock 0 1 2 3 4 5 50 mg $598 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4223701
Biological Activity
4E2RCat is a small molecule inhibitor of eIF4E-eIF4G interaction with IC50 of 13.5 uM in TR-FRET-based assay.
Physicochemical Properties
M.Wt
455.9339
Formula
C22H14ClNO4S2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: 15.5 mg/mL
Chemical Name/SMILES
Benzoic acid, 2-chloro-5-[5-[[4-oxo-3-(phenylmethyl)-2-thioxo-5-thiazolidinylidene]methyl]-2-furanyl]-
References
1. Cencic R, et al. J Virol
2. Cencic R, et al. Proc Natl Acad Sci U S A
3. Bhat M, et al. Nat Rev Drug Discov
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