AAK1 inhibitor 25A |CAS 2634715-17-4 Probechem Biochemicals

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Chemical Structure : AAK1 inhibitor 25A

AAK1 inhibitor 25A

Catalog No.: PC-35961Not For Human Use, Lab Use Only.

AAK1 inhibitor 25A is a potent, selective inhibitor of AAK1 and the closely related kinase BMP2K with Ki of 8 nM (AAK1).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

AAK1 inhibitor 25A is a potent, selective inhibitor of AAK1 and the closely related kinase BMP2K with Ki of 8 nM (AAK1).
AAK1 inhibitor 25A displays selectivity over the other members of the subfamily, Numb-associated kinases GAK and STK16, in a TR-FRET binding displacement assay.
AAK1 inhibitor 25A binds to BMP2K in live HEK293T cells with an IC50 of 602 nM.

Physicochemical Properties

M.Wt	396.465
Formula	C20H20N4O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(6-(3-(cyclopropanesulfonamido)phenyl)-1H-indazol-3-yl)cyclopropanecarboxamide

References

1. Agajanian MJ, et al. Cell Rep. 2019 Jan 2;26(1):79-93.e8.

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