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Chemical Structure : ABT-239
CAS No.: 460746-46-7
Catalog No.: PC-42908Not For Human Use, Lab Use Only.
ABT-239 is a potent and selective Histamine H3 receptor antagonist with Ki of 0.1-5.8 nM (human, rat H3).
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $98 | In stock | |
| 10 mg | $158 | In stock | |
| 25 mg | $278 | In stock | |
| 50 mg | $478 | In stock | |
| 100 mg | Get quote |
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ABT-239 is a potent and selective Histamine H3 receptor antagonist with Ki of 0.1-5.8 nM (human, rat H3).
ABT-239 exhibits 1000-fold selectivity versus H1, H2 and H4.
ABT-239 exhibits excellent pharmacokinetic and metabolic properties across species and good oral bioavailability.
| M.Wt | 330.4229 | |
| Formula | C22H22N2O | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 3.3 mg/mL |
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| Chemical Name/SMILES |
Benzonitrile, 4-[2-[2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl]-5-benzofuranyl]- |
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1. Cowart M, et al. J Med Chem. 2005 Jan 13;48(1):38-55.
2. Esbenshade TA, et al. J Pharmacol Exp Ther. 2005 Apr;313(1):165-75.
3. Bhowmik M, et al. Brain Res. 2014 Sep 18;1581:129-40.
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