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ACR-917

Chemical Structure : ACR-917

CAS No.: 2286564-50-7

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ACR-917 (ACR917)

Catalog No.: PC-28592Not For Human Use, Lab Use Only.

ACR-917 is a covalent small molecule inhibitor of Rho family GTPase RhoA protein by covalent modification of Cys107, inhibits RhoA C190S nucleotide exchange with IC50 of 46 uM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

ACR-917 is a covalent small molecule inhibitor of Rho family GTPase RhoA protein by covalent modification of Cys107, inhibits RhoA C190S nucleotide exchange with IC50 of 46 uM.

Physicochemical Properties

M.Wt 331.17
Formula C15H11BrN2O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1-(8-bromobenzo[f]pyrido[2,3-b][1,4]oxazepin-5(6H)-yl)prop-2-en-1-one

References

1. Muhammad S Hussain, et al. ACS Chem Neurosci. 2023 Jul 19;14(14):2509-2516.

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