ACT-1016-0707

Chemical Structure : ACT-1016-0707

Catalog No.: PC-21751Not For Human Use, Lab Use Only.

ACT-1016-0707 is a potent, selective, and orally active lysophosphatidic acid receptor subtype 1 receptor (LPA1 receptor, LPAR1) antagonist with IC50 of 3.1 nM, highly selective over LPAR2 or LPAR3.

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Biological Activity

ACT-1016-0707 is a potent, selective, and orally active lysophosphatidic acid receptor subtype 1 receptor (LPA1 receptor, LPAR1) antagonist with IC50 of 3.1 nM, highly selective over LPAR2 or LPAR3.
ACT-1016-0707 suppressed the LPA-induced vascular leakage at a p.o. dose of 30 mg/kg.

Physicochemical Properties

M.Wt	438.93
Formula	C19H23ClN4O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(6-Chloro-4-methoxypyridin-3-yl)-3-(2-isopropylphenyl)-1-sulfamoylazetidine-3-carboxamide

References

1. Lescop C, et al. J Med Chem. 2024 Feb 13. doi: 10.1021/acs.jmedchem.3c01827.

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ACT-1016-0707

Biological Activity

Physicochemical Properties

References

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