Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.

You are here:Home-Chemical Inhibitors & Agonists-GPCR-Prostaglandin Receptor-AH6809
AH6809

Chemical Structure : AH6809

CAS No.: 33458-93-4

AH6809 (AH-6809)

Catalog No.: PC-42574Not For Human Use, Lab Use Only.

AH6809 is a xanthone derivative that fuctions as an EP and DP receptor antagonist with Ki of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively.

Packing Price Stock Quantity
10 mg $128 In stock
25 mg $218 In stock
50 mg $358 In stock
100 mg $528 In stock
250 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

AH6809 is a xanthone derivative that fuctions as an EP and DP receptor antagonist with Ki of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively.
AH6809 blocks the PGE2-induced accumulation of cAMP in COS cells transfected with the human EP2 receptor。
AH6809 is an effective antagonist antiaggregatory actions of PGD2, but not PGI2, with EC50 50 uM in whole human platelet.

Physicochemical Properties

M.Wt 298.2901
Formula C17H14O5
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

9H-Xanthene-2-carboxylic acid, 6-(1-methylethoxy)-9-oxo-

References

1. Armstrong RA, et al. Br J Pharmacol. 1986 Mar;87(3):543-51.

2. Woodward DF, et al. Biochem Pharmacol. 1995 Nov 9;50(10):1731-3.

3. Keery RJ, et al. Br J Pharmacol. 1988 Jul;94(3):745-54.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: