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ALB-127158

Chemical Structure : ALB-127158

CAS No.: 1173154-32-9

ALB-127158 (ALB-127158(a), ALB127158A, CSTI-100)

Catalog No.: PC-61531Not For Human Use, Lab Use Only.

ALB-127158 is a potent (IC50=7 nM), selective, non-peptide antagonist of MCHR1 (Melanin-concentrating hormone receptor 1) for treatment of obesity..

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    ALB-127158 is a potent (IC50=7 nM), selective, non-peptide antagonist of MCHR1 (Melanin-concentrating hormone receptor 1) for treatment of obesity.

    Physicochemical Properties

    M.Wt 404.45
    Formula C23H21FN4O2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    4-[(5-Fluoro-2-pyridinyl)methoxy]-1-(2,3,4,5-tetrahydro-5-methyl-1H-pyrido[4,3-b]indol-7-yl)-2(1H)-pyridinone

    References

    1. Moore NA, et al. Neurobiol Dis. 2014 Jan;61:47-54.

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