AM-5262 |CAS:1222088-90-5 Probechem Biochemicals

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Chemical Structure : AM-5262

AM-5262 (AM5262)

Catalog No.: PC-63042Not For Human Use, Lab Use Only.

AM-5262 is a potent full GPR40 (FFA1) agonist with EC50 of 81 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

AM-5262 is a potent full GPR40 (FFA1) agonist with EC50 of 81 nM.
AM-5262 shows improved rat PK profile and general selectivity profile, enhances glucose stimulated insulin secretion (mouse and human islets) and improves glucose homeostasis in vivo (OGTT in HF/STZ mice) when compared to AM-1638.

Physicochemical Properties

M.Wt	514.637
Formula	C33H35FO4
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(1R,2R)-6'-((2-((R)-2,2-dimethylcyclopentyl)-2'-fluoro-5'-methoxy-[1,1'-biphenyl]-4-yl)methoxy)-2',3'-dihydrospiro[cyclopropane-1,1'-indene]-2-carboxylic acid

References

1. Wang Y, et al. ACS Med Chem Lett. 2013 May 7;4(6):551-5.

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AM-5262 (AM5262)

Biological Activity

Physicochemical Properties

References

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