APD916 (APD-916)

Chemical Structure : APD916

Catalog No.: PC-61562Not For Human Use, Lab Use Only.

APD916 is a potent and selective antagonist of the H3 receptor with Ki of 0.7 nM for rH3R.

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Biological Activity

APD916 is a potent and selective antagonist of the H3 receptor with Ki of 0.7 nM for rH3R.
APD916 increases wakefulness in rodents as measured by polysomnography with a duration of effect consistent with its pharmacokinetic properties.

Physicochemical Properties

M.Wt	401.565
Formula	C23H31NO3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-1-(2-(4'-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl)-2-methylpyrrolidine

References

1. Semple G, et al. Bioorg Med Chem Lett. 2012 Jan 1;22(1):71-5.

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APD916 (APD-916)

Biological Activity

Physicochemical Properties

References

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