APJ agonist 47

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Chemical Structure : APJ agonist 47

Catalog No.: PC-38748Not For Human Use, Lab Use Only.

APJ agonist 47 is a potent and selective, orally active apelin receptor (APJ) agonist EC50 of 6.5 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

APJ agonist 47 is a potent and selective, orally active apelin receptor (APJ) agonist EC50 of 6.5 nM.
APJ agonist 47 has vastly reduced brain penetration and is devoid of significant off-target liability.
APJ agonist 47 is suitable for in vivo studies of APJ in peripheral tissues after oral administration.

Physicochemical Properties

M.Wt	566.581
Formula	C26H31F5N8O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-1-cyclopentyl-N-(4-(3,3-difluoropiperidin-1-yl)-1-(1H-tetrazol-5-yl)butan-2-yl)-5-(2-(trifluoromethyl)phenyl)-1H-pyrazole-3-carboxamide

References

1. Sanju Narayanan, et al. Bioorg Med Chem. 2022 May 6;66:116789.

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APJ agonist 47

Biological Activity

Physicochemical Properties

References

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