Chemical Structure : APJ agonist 47
Catalog No.: PC-38748Not For Human Use, Lab Use Only.
APJ agonist 47 is a potent and selective, orally active apelin receptor (APJ) agonist EC50 of 6.5 nM.
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APJ agonist 47 is a potent and selective, orally active apelin receptor (APJ) agonist EC50 of 6.5 nM.
APJ agonist 47 has vastly reduced brain penetration and is devoid of significant off-target liability.
APJ agonist 47 is suitable for in vivo studies of APJ in peripheral tissues after oral administration.
M.Wt | 566.581 | |
Formula | C26H31F5N8O | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Sanju Narayanan, et al. Bioorg Med Chem. 2022 May 6;66:116789.
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