Chemical Structure : ARC 239 dihydrochloride
CAS No.:
55974-42-0
ARC 239 dihydrochloride
(ARC-239;ARC239)
Catalog No. : PC-60704Not For Human Use, Lab Use Only.
ARC 239 dihydrochloride is a potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-6070401
Biological Activity
ARC 239 dihydrochloride is a potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors.
Physicochemical Properties
M.Wt
480.43
Formula
C24H29N3O3.2HCl
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
2-[2-(4-(2-Methoxyphenyl)piperazin-1-yl)ethyl]-4,4-dimethyl-1,3-(2H,4H)-isoquinolindione dihydrochloride
References
1. Mouillé P, et al. J Cardiovasc Pharmacol. 1980;2(2):175-91.
2. Bylund D, et al. J Pharmacol Exp Ther. 1988 May;245(2):600-7.
3. Bylund DB, et al. J Pharmacol Exp Ther. 1989 Nov;251(2):640-4.
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