AR NTD inhibitor 16

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Chemical Structure : AR NTD inhibitor 16

CAS No.: 3016437-05-8

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Catalog No.: PC-21578Not For Human Use, Lab Use Only.

AR NTD inhibitor 16 is a small molecule inhibitor of androgen receptor N-terminal domain (AR NTD) with IC50 of 0.12 uM in VCaP cell-based GRE2-luciferase reporter gene assays.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

AR NTD inhibitor 16 is a small molecule inhibitor of androgen receptor N-terminal domain (AR NTD) with IC50 of 0.12 uM in VCaP cell-based GRE2-luciferase reporter gene assays.
AR NTD inhibitor 16 is more potent than known AR-NTD AF1 binder EPI-001 (IC50=37.4 μM).
AR NTD inhibitor 16 is a tool compound to investigate the pharmacology and engagement of the AR NTD.

Physicochemical Properties

M.Wt	297.38
Formula	C16H15N3OS
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	Benzamide, 3-(1-methyl-1H-indazol-5-yl)-4-(methylthio)-

References

1. Martyn C Henry, et al. ACS Med Chem Lett. 2023 Nov 17;14(12):1800-1806.

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