ASP8302 | M3 PAM | Probechem Biochemicals

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Chemical Structure : ASP8302

ASP8302 (ASP-8302, ASP 8302)

Catalog No.: PC-72280Not For Human Use, Lab Use Only.

ASP8302 (ASP 8302) is a potent, selective, positive allosteric modulator (PAM) of muscarinic M3 receptor.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

ASP8302 (ASP 8302) is a potent, selective, positive allosteric modulator (PAM) of muscarinic M3 receptor.
Threonine 230 (Thr 230) is the amino acid essential for the PAM effect of ASP8302.

Physicochemical Properties

M.Wt	590.158
Formula	C26H32ClN7O3S2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-[(2S)-4-(5-{[4-(4-chlorothiophen-2-yl)-5-{[(2R)-2-methylpyrrolidin-1-yl]methyl}-1,3-thiazol-2-yl]carbamoyl}pyrazin-2-yl)-2-methylpiperazin-1-yl]propanoic acid

References

1. Okimoto R, et al. J Pharmacol Exp Ther. 2021 Oct;379(1):64-73.

2. Okimoto R, et al. Low Urin Tract Symptoms. 2022 Feb 12.

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ASP8302 (ASP-8302, ASP 8302)

Biological Activity

Physicochemical Properties

References

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