Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.
Chemical Structure : AZ12204657
Catalog No.: PC-35910Not For Human Use, Lab Use Only.
AZ12204657 (AZ-12204657) small-molecule GPR44 antagonist, displaces the binding of [3H]PGD2 from membranes of HEK293 cells transfected with human recombinant GPR44 with IC50 of 2.5 nM.
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
AZ12204657 (AZ-12204657) is a small-molecule GPR44 antagonist, displaces the binding of [3H]PGD2 from membranes of HEK293 cells transfected with human recombinant GPR44 with IC50 of 2.5 nM.
[11C]AZ12204657 is a potential PET radioligand for the beta cell-restricted protein GPR44.
| M.Wt | 405.242 | |
| Formula | C16H14Cl2O6S | |
| Appearance | Solid | |
| Storage |
|
|
| Solubility |
10 mM in DMSO |
|
1. Eriksson O, et al. Diabetes. 2018 Feb;67(2):182-192.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright
