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Chemical Structure : Asenapine maleate
CAS No.: 85650-56-2
Catalog No.: PC-42808Not For Human Use, Lab Use Only.
Asenapine maleate (Org 5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors.
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|---|---|---|---|
| 50 mg | $80 | In stock | |
| 100 mg | $112 | In stock | |
| 200 mg | $192 | In stock | |
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Asenapine maleate (Org 5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors; shows much lower affinity (pKi<5) for muscarinic receptor; behaves as a potent antagonist 5-HT receptors (5-HT2A pKB=9.0), dopaime and adrenoceptors; shows strong antipsychotic potential in vivo.
Schizophrenia
Approved
| M.Wt | 401.8402 | |
| Formula | C21H20ClNO5 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
1H-Dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, 5-chloro-2,3,3a,12b-tetrahydro-2-methyl-, (3aR,12bR)-rel-, (2Z)-2-butenedioate (1:1) |
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1. Room P, et al. Eur J Pharmacol. 1991 Dec 3;205(3):233-40.
2. Broekkamp CL, et al. Arzneimittelforschung. 1990 May;40(5):544-9.
3. Psychopharmacology (Berl). 2008 Feb;196(3):417-29.
4. Shahid M, et al. J Psychopharmacol. 2009 Jan;23(1):65-73.
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