Chemical Structure : Atipamezole hydrochloride
CAS No.:
104075-48-1
Atipamezole hydrochloride
(MPV-1248 hydrochloride;MPV1248 hydrochloride;MPV 1248 hydrochloride)
Catalog No. : PC-43011Not For Human Use, Lab Use Only.
Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4301101
Biological Activity
Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM; reverses the effects of the sedative dexmedetomidine and medetomidine as a veterinary drug.
Alcoholism
Phase 1 Discontinued
Physicochemical Properties
M.Wt
248.7512
Formula
C14H17ClN2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 47 mg/mL
Chemical Name/SMILES
1H-Imidazole, 5-(2-ethyl-2,3-dihydro-1H-inden-2-yl)-, hydrochloride (1:1)
References
1. Pertovaara A, et al. CNS Drug Rev. 2005 Autumn;11(3):273-88.
2. Scheinin H, et al. Eur J Pharmacol. 1988 Jun 22;151(1):35-42.
3. Scheinin H, et al. Eur J Pharmacol. 1986 Sep 23;129(1-2):113-21.
4. Karhuvaara S, et al. Br J Clin Pharmacol. 1990 Jul;30(1):97-106.
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