You are here:Home-Chemical Inhibitors & Agonists-Metabolic Enzyme/Protease-Phosphodiesterase (PDE)-Avanafil
Avanafil

Chemical Structure : Avanafil

CAS No.: 330784-47-9

Avanafil (TA1790;TA 1790;TA-1790)

Catalog No.: PC-45440Not For Human Use, Lab Use Only.

A potent and highly selective PDE5 inhibitor (IC50=5.2 nM) for erectile dysfunction.

Packing Price Stock Quantity
100 mg $76 In stock
500 mg $112 In stock

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

A potent and highly selective PDE5 inhibitor (IC50=5.2 nM) for erectile dysfunction; shows no significant effect on PDE1, PDE6 and PDE11.

Sexual Dysfunction

Approved

Physicochemical Properties

M.Wt 483.9507
Formula C23H26ClN7O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

5-Pyrimidinecarboxamide, 4-[[(3-chloro-4-methoxyphenyl)methyl]amino]-2-[(2S)-2-(hydroxymethyl)-1-pyrrolidinyl]-N-(2-pyrimidinylmethyl)-

References

1. Kotera J, et al. J Urol. 2012 Aug;188(2):668-74.

2. Limin M, et al. Expert Opin Investig Drugs. 2010 Nov;19(11):1427-37.

3. Wang R, et al. J Sex Med. 2012 Aug;9(8):2122-9.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: