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BAY1316957

Chemical Structure : BAY1316957

CAS No.: 1613264-40-6

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BAY1316957 (BAY 1316957)

Catalog No.: PC-36057Not For Human Use, Lab Use Only.

BAY1316957 (BAY 1316957) is a highly potent, selective, orally available human prostaglandin E2 receptor subtype 4 (hEP4-R) antagonist with IC50 of 15.3 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

BAY1316957 (BAY 1316957) is a highly potent, selective, orally available human prostaglandin E2 receptor subtype 4 (hEP4-R) antagonist with IC50 of 15.3 nM.
BAY1316957 significantly reduced pain related paw withdrawal behavior in the rat upon mechanical stimulation of the dmPGE2 treated hind paw.

Physicochemical Properties

M.Wt 441.531
Formula C27H27N3O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
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Solubility

DMSO: 100 mg/mL
Chemical Name/SMILES

2-(9-Ethyl-6-methyl-9H-carbazol-3-yl)-1-(2-methoxyethyl)-4-methyl-1H-benzimidazole-5-carboxylic acid

References

1. Bäurle S, et al. J Med Chem. 2019 Feb 1. doi: 10.1021/acs.jmedchem.8b01862.

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