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Chemical Structure : BCL6 inhibitor 8c
CAS No.: 2130878-25-8
Catalog No.: PC-61016Not For Human Use, Lab Use Only.
TP-021 (BCL6 inhibitor 8c) is a potent, in vivo-active BCL6 inhibitor with IC50 of 0.1 uM in ELISA assays.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $198 | In stock | |
| 10 mg | $298 | In stock | |
| 25 mg | $498 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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TP-021 (BCL6 inhibitor 8c) is a potent, in vivo-active BCL6 inhibitor with IC50 of 0.1 uM in ELISA assays.
BCL6 inhibitor 8c exhibits good cellular BCL6BTB/ BCoR PPI inhibitory activity in the submicromolar range (M2H IC50=0.72 uM).
BCL6 inhibitor 8c showed a good pharmacokinetic profile, which is acceptable for both in vitro and in vivo studies.
| M.Wt | 417.846 | |
| Formula | C20H20ClN3O5 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
6-((2-Chloro-4-nitro-5-((tetrahydro-2H-pyran-4-yl)oxy)phenyl)amino)-3,4-dihydroquinolin-2(1H)-one |
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1. Yasui T, et al. Bioorg Med Chem. 2017 Sep 1;25(17):4876-4886.
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