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Chemical Structure : BD-1047 dihydrobromide
CAS No.: 138356-21-5
Catalog No.: PC-63071Not For Human Use, Lab Use Only.
BD-1047 dihydrobromide is a potent, selecitve Sigma 1 receptor (σ1) antagonist with Ki of 0.93 nM.
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|---|---|---|---|
| 10 mg | $88 | In stock | |
| 25 mg | $148 | In stock | |
| 50 mg | $238 | In stock | |
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BD-1047 dihydrobromide is a potent, selecitve Sigma 1 receptor (σ1) antagonist with Ki of 0.93 nM.
BD-1047 displays 50-fold weaker affinity for sigma 2 receptor, and 100-fold selectivity over opiate, phencyclidine, muscarinic, dopamine, adrenoceptor and 5-HT receptors.
BD-1047 attenuates the dystonia induced by DTG and haloperidol in rats.
| M.Wt | 437.041 | |
| Formula | C13H22Br2Cl2N2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
N-(2-(3,4-Dichlorphenyl)ethyl)-N,N',N'-trimethyl-1,2-ethandiamine dihydrobromide |
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1. Matsumoto RR, et al. Eur J Pharmacol. 1995 Jul 14;280(3):301-10.
2. Zambon AC, et al. Eur J Pharmacol. 1997 Apr 11;324(1):39-47.
3. Roh DH, et al. Anesthesiology. 2008 Nov;109(5):879-89.
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