BI-4916 | PHGDH inhibitor | Probechem Biochemicals

Chemical Structure : BI-4916

Catalog No.: PC-72879Not For Human Use, Lab Use Only.

BI-4916 (BI-4916) is the prodrug of BI-4924, which is a potent, selective NADH/NAD+-competitive PHGDH inhibitor with IC50 of 2 nM.

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Biological Activity

BI-4916 (BI-4916) is the prodrug of BI-4924, which is a potent, selective NADH/NAD+-competitive PHGDH inhibitor with IC50 of 2 nM.

M.Wt	527.413
Formula	C23H24Cl2N2O6S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Ethyl 2-{4-[(1S)-1-[(4,5-dichloro-1,6-dimethyl-1H-indol-2-yl)formamido]-2-hydroxyethyl]benzenesulfonyl}acetate

1. Harald Weinstabl, et al. J Med Chem. 2019 Sep 12;62(17):7976-7997.