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BI-4924

Chemical Structure : BI-4924

CAS No.: 2244452-09-1

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BI-4924 (BI 4924)

Catalog No.: PC-72878Not For Human Use, Lab Use Only.

BI-4924 (BI 4924) is a potent, selective NADH/NAD+-competitive PHGDH inhibitor with IC50 of 2 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

BI-4924 (BI 4924) is a potent, selective NADH/NAD+-competitive PHGDH inhibitor with IC50 of 2 nM.
BI-4924 displays high selectivity against the majority of other dehydrogenase targets.

Physicochemical Properties

M.Wt 499.359
Formula C21H20Cl2N2O6S
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-{4-[(1S)-1-[(4,5-Dichloro-1,6-dimethyl-1H-indol-2-yl)formamido]-2-hydroxyethyl]benzenesulfonyl}acetic acid

References

1. Harald Weinstabl, et al. J Med Chem. 2019 Sep 12;62(17):7976-7997.

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