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Chemical Structure : BI 186908
Catalog No.: PC-61512Not For Human Use, Lab Use Only.
A potent and selective MCH-R1 antagonist with IC50 of 22 nM, Ki of 14 nM.
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A potent and selective MCH-R1 antagonist with IC50 of 22 nM, Ki of 14 nM; significantly reduces body weight comparable to sibutramine in a 4 week diet-induced obesity model in rats, possesses favorable DMPK and CMC properties.
| M.Wt | 422.485 | |
| Formula | C23H26N4O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Oost T, et al. Bioorg Med Chem Lett. 2015 Aug 15;25(16):3275-80.
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