BMS-242 | PD-1/PD-L1 inhibitor | Probechem Biochemicals

Chemical Structure : BMS-242

Catalog No.: PC-70032Not For Human Use, Lab Use Only.

BMS-242 is a potent PD-1/PD-L1 interaction inhibitor with IC50 of 6-100 nM in a homogenous time-resolved fluorescence binding assay.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

BMS-242 is a potent PD-1/PD-L1 interaction inhibitor with IC50 of 6-100 nM in a homogenous time-resolved fluorescence binding assay.

M.Wt	449.591
Formula	C28H35NO4
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-2-((2,6-dimethoxy-4-((2-methyl-[1,1'-biphenyl]-3-yl)methoxy)benzyl)amino)-3-methylbutan-1-ol

1. Guzik K, et al. J Med Chem. 2017 Jul 13;60(13):5857-5867.

2. Zak KM, et al. Oncotarget. 2016 May 24;7(21):30323-35.

3. Chupak, L.S., and Zheng, X. Compounds useful as immunomodulators. PCT/US2014/053695, (2015).