BMS-582949 | p38 MAPK inhibitor | Probechem Biochemicals

Chemical Structure : BMS-582949

CAS No.: 623152-17-0

BMS-582949 (BMS 582949)

Catalog No.: PC-21600Not For Human Use, Lab Use Only.

BMS-582949 is a potent, selective and orally active p38α MAP kinase inhibitor with IC50 of 13 nM, exhibits significant inhibition of TNFα release in hPBMC with IC50 of 50 nM.

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5 mg	$158	In stock
10 mg	$248	In stock
25 mg	$398	In stock
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Biological Activity

BMS-582949 is a potent, selective and orally active p38α MAP kinase inhibitor with IC50 of 13 nM, exhibits significant inhibition of TNFα release in hPBMC with IC50 of 50 nM.

Physicochemical Properties

M.Wt	406.49
Formula	C22H26N6O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	4-((5-(Cyclopropylcarbamoyl)-2-methylphenyl)amino)-5-methyl-N-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide

References

1. Liu C, et al. J Med Chem. 2010 Sep 23;53(18):6629-39.

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BMS-582949 (BMS 582949)

Biological Activity

Physicochemical Properties

References

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