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Chemical Structure : BMS-819881
Catalog No.: PC-61121Not For Human Use, Lab Use Only.
A potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.
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BMS-819881 is a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.
BMS-819881 effectively blocks MCH stimulated Ca+2 mobilization in heterologous cells overexpressing MCHR1 but not the cells expressing MCHR2 at 10 uM.
BMS-819881 shows potential for treatment of obesity.
| M.Wt | 468.952 | |
| Formula | C24H21ClN2O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Washburn WN, et al. J Med Chem. 2014 Sep 25;57(18):7509-22.
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