BMS-819881 | MCHR1 inhibitor | Probechem Biochemicals

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Chemical Structure : BMS-819881

BMS-819881 (BMS819881)

Catalog No.: PC-61121Not For Human Use, Lab Use Only.

A potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

BMS-819881 is a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.
BMS-819881 effectively blocks MCH stimulated Ca+2 mobilization in heterologous cells overexpressing MCHR1 but not the cells expressing MCHR2 at 10 uM.
BMS-819881 shows potential for treatment of obesity.

Physicochemical Properties

M.Wt	468.952
Formula	C24H21ClN2O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-6-(4-chlorophenyl)-3-(4-(2-cyclopropyl-2-hydroxyethoxy)-3-methoxyphenyl)-thieno[3,2-d]pyrimidin-4(3H)-one

References

1. Washburn WN, et al. J Med Chem. 2014 Sep 25;57(18):7509-22.

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BMS-819881 (BMS819881)

Biological Activity

Physicochemical Properties

References

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