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BMS-830216

Chemical Structure : BMS-830216

CAS No.: 1197420-06-6

BMS-830216 (BMS830216)

Catalog No.: PC-61122Not For Human Use, Lab Use Only.

The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    BMS-830216 is the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.
    BMS-830216 shows potential for treatment of obesity.

    Physicochemical Properties

    M.Wt 548.931
    Formula C24H22ClN2O7PS
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    (R)-2-(4-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-2-methoxyphenoxy)-1-cyclopropylethyl dihydrogen phosphate

    References

    1. Washburn WN, et al. J Med Chem. 2014 Sep 25;57(18):7509-22.

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