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BMS-986121

Chemical Structure : BMS-986121

CAS No.: 313671-26-0

BMS-986121 (BMS986121)

Catalog No.: PC-22779Not For Human Use, Lab Use Only.

BMS-986121 is a positive allosteric modulator of μ-opioid receptor (MOR) with EC50 of 1 uM for increased β-arrestin recruitment by 20 nM endomorphin-I.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

BMS-986121 is a positive allosteric modulator of μ-opioid receptor (MOR) with EC50 of 1 uM for increased β-arrestin recruitment by 20 nM endomorphin-I.

Physicochemical Properties

M.Wt 366.22
Formula C15H9Cl2N3O2S
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

2-Thiazolamine, N-(2,6-dichlorophenyl)-4-(4-nitrophenyl)-

References

1. Bisignano P, et al. J Chem Inf Model. 2015 Sep 28;55(9):1836-43.

2. Burford NT, et al. Proc Natl Acad Sci U S A. 2013 Jun 25;110(26):10830-5.

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