Chemical Structure : BMS-986124
Catalog No.: PC-22781Not For Human Use, Lab Use Only.
BMS-986124 is a small molecule silent allosteric modulator (SAM) of μ-opioid receptor (MOR), blocks the effects of the MOR positive allosteric modulator BMS-986122, but does not affect binding or activities of orthosteric MOR agonists such as endomorphin-I or DAMGO.
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BMS-986124 is a small molecule silent allosteric modulator (SAM) of μ-opioid receptor (MOR), blocks the effects of the MOR positive allosteric modulator BMS-986122, but does not affect binding or activities of orthosteric MOR agonists such as endomorphin-I or DAMGO.
M.Wt | 448.77 | |
Formula | C16H15BrClNO3S2 | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Kaneko S, et al. Nat Commun. 2024 May 13;15(1):3544.
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