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BMS-986124

Chemical Structure : BMS-986124

CAS No.: 1447968-71-9

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BMS-986124 (BMS986124)

Catalog No.: PC-22781Not For Human Use, Lab Use Only.

BMS-986124 is a small molecule silent allosteric modulator (SAM) of μ-opioid receptor (MOR), blocks the effects of the MOR positive allosteric modulator BMS-986122, but does not affect binding or activities of orthosteric MOR agonists such as endomorphin-I or DAMGO.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

BMS-986124 is a small molecule silent allosteric modulator (SAM) of μ-opioid receptor (MOR), blocks the effects of the MOR positive allosteric modulator BMS-986122, but does not affect binding or activities of orthosteric MOR agonists such as endomorphin-I or DAMGO.

Physicochemical Properties

M.Wt 448.77
Formula C16H15BrClNO3S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-(4-Bromo-2-methoxyphenyl)-3-[(4-chlorophenyl)sulfonyl]-thiazolidine

References

1. Kaneko S, et al. Nat Commun. 2024 May 13;15(1):3544.

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