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Chemical Structure : BMS-986187
CAS No.: 684238-37-7
Catalog No.: PC-63082Not For Human Use, Lab Use Only.
BMS-986187 is a novel potent, positive allosteric modulator of δ-opioid receptor (DOR) with EC50 of 30 nM, 100-fold selectivity over μ-opioid receptor.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $88 | In stock | |
| 10 mg | $138 | In stock | |
| 25 mg | $228 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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BMS-986187 is a novel potent, positive allosteric modulator of δ-opioid receptor (DOR) with EC50 of 30 nM, 100-fold selectivity over μ-opioid receptor.
| M.Wt | 470.609 | |
| Formula | C31H34O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
3,4,5,6,7,9-Hexahydro-3,3,6,6-tetramethyl-9-[4-[(2-methylphenyl)methoxy]phenyl]-1H-xanthene-1,8(2H)-dione |
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1. Livingston KE, et al. Mol Pharmacol. 2018 Feb;93(2):157-167.
2. Shang Y, et al. ACS Chem Biol. 2016 May 20;11(5):1220-9.
3. Burford NT, et al. J Med Chem. 2015 May 28;58(10):4220-9.
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