Chemical Structure : BMS-986205
CAS No.: 1923833-60-6
Catalog No.: PC-60068Not For Human Use, Lab Use Only.
BMS-986205 (Linrodostat, F-001287, ONO-7701) is a novel potent, selective and orally available IDO1 inhibitor with IC50 of 1.1 nM in cell-based assays.
Packing | Price | Stock | Quantity |
---|---|---|---|
5 mg | $118 | In stock | |
25 mg | $348 | In stock | |
100 mg | $988 | In stock | |
500 mg | Get quote |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
BMS-986205 (Linrodostat, F-001287, ONO-7701) is a novel potent, selective and orally available IDO1 inhibitor with IC50 of 1.1 nM in cell-based assays; has no inhibitory activity on TDO, potently inhibits kynurenine (kyn) production in IDO1-HEK293 cells with IC50 of 1.1 nM; shows potential with superior PD properties and support further evaluation in combination with vivo.
Skin Cancer
Phase 2 Clinical
M.Wt | 410.912 | |
Formula | C24H24ClFN2O | |
Appearance | Solid | |
Storage |
|
|
Solubility |
10 mM in DMSO |
|
Chemical Name/SMILES |
(2R)-N-(4-Chlorophenyl)-2-[cis-4-(6-fluoro-4-quinolinyl)cyclohexyl]propanamide |
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright