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BMS 986188

Chemical Structure : BMS 986188

CAS No.: 1776115-10-6

BMS 986188 (BMS986188)

Catalog No.: PC-38532Not For Human Use, Lab Use Only.

BMS 986188 is a potent, selective positive allosteric modulator of δ-opioid receptor with EC50 of 0.05 uM in β-arrestin recruitment assays, no significant acitivity against μ-opioid receptors.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

BMS 986188 is a potent, selective positive allosteric modulator of δ-opioid receptor with EC50 of 0.05 uM in β-arrestin recruitment assays, no significant acitivity against μ-opioid receptors.

Physicochemical Properties

M.Wt 535.5
Formula C30H31BrO4
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

9-[4-[(2-bromophenyl)methoxy]phenyl]-3,4,5,6,7,9-hexahydro-3,3,6,6-tetramethyl-1H-xanthene-1,8(2H)-dione

References

1. Burford NT, et al. J Med Chem. 2015 May 28;58(10):4220-9.

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