BPR1M492

Chemical Structure : BPR1M492

Catalog No.: PC-27320Not For Human Use, Lab Use Only.

BPR1M492 is a potent, selective, fast-acting μ-opioid receptor (MOR) agonist with EC50 of 4 nM in FLIPR Ca2+ assays, Emax=92.7%.

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Biological Activity

BPR1M492 is a potent, selective, fast-acting μ-opioid receptor (MOR) agonist with EC50 of 4 nM in FLIPR Ca2+ assays, Emax=92.7%.
BPR1M492 demonstrates potent in vivo antinociception at 0.027 mg/kg, offering rapid pain relief within 5 min of subcutaneous injection.
BPR1M492 produced markedly milder withdrawal symptoms than TRV130 in mice.

Physicochemical Properties

M.Wt	320.44
Formula	C21H24N2O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	1H-Indene-2-carboxamide, 2,3-dihydro-N-[[(3R)-1,2,3,4-tetrahydro-2-methyl-3-isoquinolinyl]methyl]-

References

1. Po-Wei Chang, et al. J Med Chem. 2026 Jun 11;69(11):13222-13247.

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BPR1M492

Biological Activity

Physicochemical Properties

References

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