Chemical Structure : BRL-44408 maleate
CAS No.:
681806-46-2
BRL-44408 maleate
(BRL44408)
Catalog No. : PC-60703Not For Human Use, Lab Use Only.
BRL-44408 maleate is a potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-6070301
Biological Activity
BRL-44408 maleate is a potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors.
Physicochemical Properties
M.Wt
331.372
Formula
C17H21N3O4
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole maleate
References
1. Kiss JP, et al. Brain Res. 1995 Mar 20;674(2):238-44.
2. Callado LF, et al. Eur J Pharmacol. 1999 Jan 29;366(1):35-9.
3. Young P, et al. Eur J Pharmacol. 1989 Sep 22;168(3):381-6.
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