Bavarostat | HDAC6 inhibitor | Probechem Biochemicals

Chemical Structure : Bavarostat

CAS No.: 2134109-20-7

Bavarostat (EKZ-001)

Catalog No.: PC-24769Not For Human Use, Lab Use Only.

Bavarostat (EKZ-001) is a potent, selective HDAC6 inhibitor with IC50 of 60 nM, 16000-fold selectivity over HDAC1, HDAC2, and HDAC3.

Packing	Price	Stock
5 mg	$98	In stock
10 mg	$148	In stock
25 mg	$258	In stock
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Biological Activity

Bavarostat (EKZ-001) is a potent, selective HDAC6 inhibitor with IC50 of 60 nM, 16000-fold selectivity over HDAC1, HDAC2, and HDAC3.
Bavarostat is used as a brain-penetrant positron emission tomography (PET) probe for imaging HDAC6 in the central nervous system.

Physicochemical Properties

M.Wt	346.45
Formula	C20H27FN2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(((Adamantan-1-ylmethyl)(methyl)amino)methyl)-3-fluoro-N-hydroxybenzamide

References

1. Wagner FF, et al. ACS Cent Sci. 2017 Sep 27;3(9):1006-1014.

2. Porter NJ, et al. J Med Chem. 2018 Sep 13;61(17):8054-8060.

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Bavarostat (EKZ-001)

Biological Activity

Physicochemical Properties

References

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