Catalog No.: PC-24453Not For Human Use, Lab Use Only.
Brexpiprazole (OPC-34712) is an atypical orally active antipsychotic agent and partial agonist of human 5-HT1A and dopamine D2L receptor with Ki of 0.12 nM and 0.3 nM, respectively.
Brexpiprazole (OPC-34712) is an atypical orally active antipsychotic agent and partial agonist of human 5-HT1A and dopamine D2L receptor with Ki of 0.12 nM and 0.3 nM, respectively. Brexpiprazole (OPC-34712) is also a 5-HT2A receptor antagonist with Ki of 0.47 nM. Brexpiprazole also shows potent antagonist activity at human noradrenergic α1B (Ki=0.17 nM) and α2C receptors (Ki=0.59 nM).
