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CAM4066

Chemical Structure : CAM4066

CAS No.: 2101206-81-7

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CAM4066 (CAM 4066, CAM-4066)

Catalog No.: PC-35184Not For Human Use, Lab Use Only.

CAM4066 (CAM-4066) is a potent and selective CK2alpha (CK2α) inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM, shows significantly improved selectivity compared to other CK2α inhibitors.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    CAM4066 (CAM-4066) is a potent and selective CK2alpha (CK2α) inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM, shows significantly improved selectivity compared to other CK2α inhibitors.
    CAM4066 inhibits CK2 activity by exploiting a pocket located outside the ATP binding site (alphaD pocket).

    Physicochemical Properties

    M.Wt 479.961
    Formula C26H26ClN3O4
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    3-(3-(3-(((2-chloro-[1,1'-biphenyl]-4-yl)methyl)amino)propanamido)propanamido)benzoic acid

    References

    1. Iegre J, et al. Chem Sci. 2018 Feb 20;9(11):3041-3049.

    2. Brear P, et al. Chem Sci. 2016 Nov 1;7(11):6839-6845.

    3. De Fusco C, et al. Bioorg Med Chem. 2017 Jul 1;25(13):3471-3482.

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