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CCT373567

Chemical Structure : CCT373567

CAS No.: 2378853-67-7

CCT373567 (CCT 373567)

Catalog No.: PC-20626Not For Human Use, Lab Use Only.

CCT373567 is a potent, selective and cell-active BCL6 inhibitor with IC50 of 2.9 nM in TR-FRET assays, and 25.9 nM in NanoBRET cellular inhibition assays.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    CCT373567 is a potent, selective and cell-active BCL6 inhibitor with IC50 of 2.9 nM in TR-FRET assays, and 25.9 nM in NanoBRET cellular inhibition assays.

    Physicochemical Properties

    M.Wt 547.00
    Formula C26H29ClF2N6O3
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    (S)-10-((5-chloro-2-((3S,5R)-3-hydroxy-5-methylpiperidin-1-yl)pyrimidin-4-yl)amino)-2-cyclopropyl-3,3-difluoro-7-methyl-1,2,3,4-tetrahydro-[1,4]oxazepino[2,3-c]quinolin-6(7H)-one

    References

    1. Alice C Harnden, et al. J Med Chem. 2023 Apr 7. doi: 10.1021/acs.jmedchem.3c00155.

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