CFT-1297 | BRD4 PROTAC | Probechem Biochemicals

Chemical Structure : CFT-1297

Catalog No.: PC-23208Not For Human Use, Lab Use Only.

CFT-1297 is a potent, selective BRD4 PROTAC degrader with DC50 of 5 nM and Dmax of 97% in HEK293T cells, targets the BD1 domain of BRD4.

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Biological Activity

CFT-1297 is a potent, selective BRD4 PROTAC degrader with DC50 of 5 nM and Dmax of 97% in HEK293T cells, targets the BD1 domain of BRD4.

M.Wt	824.43
Formula	C47H50ClN9O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-(4-(1-(7-(4-(6-(4-chlorophenyl)-1-methylspiro[benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepine-4,1'-cyclopropan]-8-yl)-1H-pyrazol-1-yl)heptyl)piperidin-4-yl)-1-oxoisoindolin-2-yl)piperidine-2,6-dione

1. Eron SJ, et al. ACS Chem Biol. 2021 Nov 19;16(11):2228-2243.