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Chemical Structure : CH5447240
Catalog No.: PC-35255Not For Human Use, Lab Use Only.
CH5447240 is a novel potent, selective, orally active hPTHR1 agonist with EC20 of 3.0 nM and EC50 of 12 nM.
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CH5447240 is a novel potent, selective, orally active hPTHR1 agonist with EC20 of 3.0 nM and EC50 of 12 nM.
CH5447240 shows excellent physicochemical properties, such as high solubility in fasted state simulated intestinal fluid and good metabolic stability in human liver microsomes.
CH5447240 demonstrates a significantly elevated serum calcium level in hypocalcemic model rats.
| M.Wt | 517.689 | |
| Formula | C26H39N5O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Nishimura Y, et al. J Med Chem. 2018 Jun 22. doi: 10.1021/acs.jmedchem.8b00182.
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