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CHF-6550

Chemical Structure : CHF-6550

CAS No.:

CHF-6550 (CHF6550)

Catalog No.: PC-22509Not For Human Use, Lab Use Only.

CHF-6550 is a potent, dual acting muscarinic M3 antagonist and β2 agonist (MABA) with pKi values of 9.3 and 10.6 for M3 and β2 receptor, respectively.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

CHF-6550 is a potent, dual acting muscarinic M3 antagonist and β2 agonist (MABA) with pKi values of 9.3 and 10.6 for M3 and β2 receptor, respectively.

Physicochemical Properties

M.Wt 734.85
Formula C42H46N4O8
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(S)-1-methylpiperidin-3-yl (R)-2-hydroxy-2-(3-(3-(4-((((R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethyl)amino)methyl)benzamido)propoxy)phenyl)-2-phenylacetate

References

1. Laura Carzaniga, et al. J Med Chem. 2024 Jun 10. doi: 10.1021/acs.jmedchem.4c00298.

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