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CK156

Chemical Structure : CK156

CAS No.:

CK156 (CK-156)

Catalog No.: PC-38745Not For Human Use, Lab Use Only.

CK156 is a potent, highly selective serine/threonine kinase 17A (DRAK1) inhibitor with Kd of 21 nM, cellular IC50 of 182 nM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

CK156 is a potent, highly selective serine/threonine kinase 17A (STK17A, DRAK1) inhibitor with Kd of 21 nM, cellular IC50 of 182 nM.
CK156 demonstrates excellent selectivity in kinomewide screens.
CK156 inhibits cell growth of glioma cells in 2D and 3D culture only at low micromolar concentrations.

Physicochemical Properties

M.Wt 395.463
Formula C21H25N5O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

References

1. Christian G Kurz, et al. J Med Chem. 2022 May 24. doi: 10.1021/acs.jmedchem.2c00173.

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