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Chemical Structure : CK156
Catalog No.: PC-38745Not For Human Use, Lab Use Only.
CK156 is a potent, highly selective serine/threonine kinase 17A (DRAK1) inhibitor with Kd of 21 nM, cellular IC50 of 182 nM.
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CK156 is a potent, highly selective serine/threonine kinase 17A (STK17A, DRAK1) inhibitor with Kd of 21 nM, cellular IC50 of 182 nM.
CK156 demonstrates excellent selectivity in kinomewide screens.
CK156 inhibits cell growth of glioma cells in 2D and 3D culture only at low micromolar concentrations.
| M.Wt | 395.463 | |
| Formula | C21H25N5O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Christian G Kurz, et al. J Med Chem. 2022 May 24. doi: 10.1021/acs.jmedchem.2c00173.
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