You are here:Home-Chemical Inhibitors & Agonists-GPCR-Oxytocin Receptor (OXTR)-Carbetocin
Carbetocin

Chemical Structure : Carbetocin

CAS No.: 37025-55-1

Carbetocin

Catalog No.: PC-45361Not For Human Use, Lab Use Only.

Carbetocin is an oxytocin (OT) analogue and potent agonist of peripheral oxytocin receptor with Ki of 7 nM.

Packing Price Stock Quantity
25 mg $98 In stock
50 mg $158 In stock
100 mg $258 In stock
250 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Carbetocin is an oxytocin (OT) analogue and potent agonist of peripheral oxytocin receptor with Ki of 7 nM.
Carbetocin shows high affinity to chimeric N-terminus (E1) of the oxytocin receptor (Ki=1.17 μM).
Carbetocin shows significant effect of treatment on the percent time spent climbing, swimming and immobile.
Carbetocin is used in obstetrics to control postpartum hemorrhage and bleeding after giving birth, particularly following Cesarean section.

Physicochemical Properties

M.Wt 988.1609
Formula C45H69N11O12S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: ≥ 31 mg/mL

Chemical Name/SMILES

Glycinamide, N-(4-mercapto-1-oxobutyl)-O-methyl-L-tyrosyl-L-isoleucyl-L-glutaminyl-L-asparaginyl-L-cysteinyl-L-prolyl-L-leucyl-, cyclic (1→5)-thioether

References

1. Stella Chaviaras, et al. Psychopharmacology (Berl). 2010 May;210(1):35-43.
2. Gerald Gimpl, et al. Eur J Pharmacol. 2005 Mar 7;510(1-2):9-16.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: