Chemical Structure : Carbetocin
CAS No.:
37025-55-1
Carbetocin
Catalog No.: PC-45361Not For Human Use, Lab Use Only.
Carbetocin is an oxytocin (OT) analogue and potent agonist of peripheral oxytocin receptor with Ki of 7 nM.
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Purity & Documentation Purity:
>98% (HPLC)
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Biological Activity
Carbetocin is an oxytocin (OT) analogue and potent agonist of peripheral oxytocin receptor with Ki of 7 nM.
Carbetocin shows high affinity to chimeric N-terminus (E1) of the oxytocin receptor (Ki=1.17 μM).
Carbetocin shows significant effect of treatment on the percent time spent climbing, swimming and immobile.
Carbetocin is used in obstetrics to control postpartum hemorrhage and bleeding after giving birth, particularly following Cesarean section.
Physicochemical Properties
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M.Wt
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988.1609
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Formula
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C45H69N11O12S
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Appearance
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Solid
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CAS No.
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Storage
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- Solide Powder
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-20 °C 12 Months; 4°C 6 Months
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- In Solvent
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-80 °C 6 Months; -20°C 6 Months
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Shipping
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Solubility
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DMSO: ≥ 31 mg/mL
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Chemical Name/SMILES
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Glycinamide, N-(4-mercapto-1-oxobutyl)-O-methyl-L-tyrosyl-L-isoleucyl-L-glutaminyl-L-asparaginyl-L-cysteinyl-L-prolyl-L-leucyl-, cyclic (1→5)-thioether
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References
1. Stella Chaviaras, et al. Psychopharmacology (Berl). 2010 May;210(1):35-43.
2. Gerald Gimpl, et al. Eur J Pharmacol. 2005 Mar 7;510(1-2):9-16.
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