Chemical Structure : Cisapride
CAS No.: 81098-60-4
Catalog No.: PC-28211Not For Human Use, Lab Use Only.
Cisapride (R 51619) is a potent, selective and orally active 5-HT4 receptor agonist with EC50 of 140 nM, is also an hERG potassium channel blocker with IC50 of 9.4 nM, inhibits voltage-dependent K(+) (Kv) channels using freshly isolated smooth muscle cells.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 50 mg | $58 | In stock | |
| 100 mg | $88 | In stock | |
| 250 mg | $128 | In stock | |
| 1 g | Get quote |
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Cisapride (R 51619) is a potent, selective and orally active 5-HT4 receptor agonist with EC50 of 140 nM, is also an hERG potassium channel blocker with IC50 of 9.4 nM, inhibits voltage-dependent K(+) (Kv) channels using freshly isolated smooth muscle cells.
| M.Wt | 465.95 | |
| Formula | C23H29ClFN3O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
rel-4-Amino-5-chloro-N-((3R,4S)-1-(3-(4-fluorophenoxy)propyl)-3-methoxypiperidin-4-yl)-2-methoxybenzamide |
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1. Kim HW, et al. Biochem Biophys Res Commun. 2016 Sep 23;478(3):1423-8.
2. Walker BD, et al. Br J Pharmacol. 1999 Sep;128(2):444-50.
3. Ueki S, et al. J Pharmacol Exp Ther. 1993 Jan;264(1):152-7.

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