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Chemical Structure : Cligosiban
CAS No.: 900510-03-4
Catalog No.: PC-61369Not For Human Use, Lab Use Only.
Cligosiban (PF-3274167) is a potent, specific oxytocin receptor antagonist with Ki of 9.5 nM, displays high selectivity over the vasopressin receptors.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $88 | In stock | |
| 25 mg | $138 | In stock | |
| 50 mg | $218 | In stock | |
| 100 mg | Get quote |
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Cligosiban (PF-3274167) is a potent, specific oxytocin receptor antagonist with Ki of 9.5 nM, displays high selectivity over the vasopressin receptors.
Cligosiban (PF-3274167) demonstrates excellent potency and selectivity, as well as promising in vivo pharmacokinetics and significantly improved aqueous solubility.
| M.Wt | 419.841 | |
| Formula | C19H19ClFN5O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
5-(3-(3-(2-chloro-4-fluorophenoxy)azetidin-1-yl)-5-(methoxymethyl)-4H-1,2,4-triazol-4-yl)-2-methoxypyridine |
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1. Vidal B, et al. Nucl Med Biol. 2017 Dec;55:1-6.
2. Brown A, et al. Bioorg Med Chem Lett. 2010 Jan 15;20(2):516-20.
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